AF6/ERBIN/SNA1 PDZ domain - Selectivity below 100 micro-molar
Recognized by the AF6, ERBIN and SNA1 PDZ domains
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| P3 |
P2 |
P1 |
P0 |
Seq. |
AF6-Kd |
ERBIN-Kd |
SNA1-Kd |
| G |
T |
F |
V |
GTFV |
9.22 |
71.09 |
91.78 |
| A |
T |
F |
V |
ATFV |
9.95 |
75.83 |
47.76 |
| E |
I |
W |
V |
EIWV |
10.33 |
30.52 |
76.51 |
| G |
T |
W |
V |
GTWV |
10.36 |
33.97 |
51.65 |
| A |
T |
W |
V |
ATWV |
11.18 |
36.23 |
26.88 |
| E |
T |
F |
V |
ETFV |
12.17 |
13.93 |
18.70 |
| E |
V |
W |
V |
EVWV |
13.43 |
20.80 |
72.70 |
| E |
F |
W |
V |
EFWV |
13.51 |
56.62 |
93.24 |
| E |
T |
W |
V |
ETWV |
13.66 |
6.66 |
10.52 |
| P |
T |
W |
V |
PTWV |
15.62 |
60.29 |
91.06 |
| E |
L |
W |
V |
ELWV |
15.82 |
73.46 |
99.36 |
| S |
T |
F |
V |
STFV |
17.35 |
56.91 |
36.18 |
| G |
S |
W |
V |
GSWV |
18.11 |
64.78 |
50.13 |
| S |
T |
W |
V |
STWV |
19.48 |
27.19 |
20.36 |
| A |
S |
W |
V |
ASWV |
19.55 |
69.09 |
26.09 |
| E |
S |
F |
V |
ESFV |
21.28 |
26.57 |
18.15 |
| E |
T |
Y |
V |
ETYV |
21.64 |
32.15 |
12.61 |
| E |
T |
L |
V |
ETLV |
23.41 |
69.99 |
16.15 |
| E |
S |
W |
V |
ESWV |
23.89 |
12.70 |
10.21 |
| E |
T |
F |
I |
ETFI |
27.89 |
62.24 |
29.08 |
| E |
I |
W |
L |
EIWL |
28.38 |
77.84 |
97.07 |
| G |
T |
W |
L |
GTWL |
28.45 |
86.65 |
65.54 |
| A |
T |
W |
L |
ATWL |
30.71 |
92.42 |
34.10 |
| E |
T |
W |
I |
ETWI |
31.32 |
29.74 |
16.37 |
| W |
T |
F |
V |
WTFV |
32.10 |
82.17 |
86.84 |
| D |
T |
F |
V |
DTFV |
32.25 |
26.12 |
54.37 |
| Q |
T |
F |
V |
QTFV |
33.31 |
76.91 |
36.81 |
| E |
T |
F |
L |
ETFL |
33.43 |
35.55 |
23.73 |
| S |
S |
W |
V |
SSWV |
34.07 |
51.85 |
19.76 |
| W |
T |
W |
V |
WTWV |
36.04 |
39.26 |
48.87 |
| D |
T |
W |
V |
DTWV |
36.22 |
12.48 |
30.60 |
| E |
V |
W |
L |
EVWL |
36.91 |
53.05 |
92.25 |
| V |
T |
F |
V |
VTFV |
37.08 |
58.41 |
35.02 |
| H |
T |
F |
V |
HTFV |
37.23 |
80.65 |
39.87 |
| T |
T |
F |
V |
TTFV |
37.39 |
65.45 |
57.74 |
| Q |
T |
W |
V |
QTWV |
37.40 |
36.75 |
20.71 |
| E |
T |
W |
L |
ETWL |
37.54 |
16.98 |
13.35 |
| E |
S |
Y |
V |
ESYV |
37.85 |
61.31 |
12.24 |
| E |
T |
W |
F |
ETWF |
41.23 |
90.38 |
38.87 |
| V |
T |
W |
V |
VTWV |
41.63 |
27.91 |
19.71 |
| H |
T |
W |
V |
HTWV |
41.81 |
38.53 |
22.44 |
| T |
T |
W |
V |
TTWV |
41.98 |
31.27 |
32.50 |
| F |
T |
F |
V |
FTFV |
42.58 |
76.78 |
54.20 |
| E |
T |
T |
V |
ETTV |
42.75 |
61.50 |
6.13 |
| I |
T |
F |
V |
ITFV |
46.62 |
68.07 |
59.61 |
| N |
T |
F |
V |
NTFV |
47.58 |
94.03 |
51.27 |
| F |
T |
W |
V |
FTWV |
47.81 |
36.68 |
30.50 |
| Y |
T |
W |
V |
YTWV |
48.88 |
54.75 |
46.04 |
| E |
I |
D |
V |
EIDV |
49.71 |
88.66 |
73.65 |
| G |
T |
D |
V |
GTDV |
49.83 |
98.69 |
49.72 |
| E |
A |
W |
V |
EAWV |
50.09 |
47.64 |
70.63 |
| I |
T |
W |
V |
ITWV |
52.36 |
32.52 |
33.55 |
| E |
H |
W |
V |
EHWV |
52.48 |
68.18 |
89.27 |
| N |
T |
W |
V |
NTWV |
53.43 |
44.93 |
28.86 |
| S |
T |
W |
L |
STWL |
53.53 |
69.36 |
25.83 |
| E |
Q |
W |
V |
EQWV |
54.70 |
58.91 |
80.13 |
| E |
S |
W |
I |
ESWI |
54.76 |
56.71 |
15.89 |
| D |
S |
F |
V |
DSFV |
56.40 |
49.81 |
52.77 |
| E |
V |
N |
V |
EVNV |
56.83 |
90.23 |
61.05 |
| M |
T |
F |
V |
MTFV |
56.93 |
90.22 |
42.29 |
| D |
T |
Y |
V |
DTYV |
57.37 |
60.26 |
36.66 |
| E |
T |
N |
V |
ETNV |
57.80 |
28.89 |
8.84 |
| E |
S |
F |
L |
ESFL |
58.46 |
67.79 |
23.03 |
| E |
T |
E |
V |
ETEV |
59.45 |
45.09 |
8.79 |
| E |
T |
Y |
L |
ETYL |
59.47 |
82.01 |
16.00 |
| E |
V |
S |
V |
EVSV |
62.30 |
77.74 |
65.01 |
| E |
T |
Q |
V |
ETQV |
62.60 |
33.81 |
9.78 |
| W |
S |
W |
V |
WSWV |
63.03 |
74.87 |
47.43 |
| D |
S |
W |
V |
DSWV |
63.34 |
23.80 |
29.70 |
| E |
T |
S |
V |
ETSV |
63.37 |
24.89 |
9.41 |
| M |
T |
W |
V |
MTWV |
63.93 |
43.11 |
23.80 |
| L |
T |
W |
V |
LTWV |
64.57 |
55.52 |
37.02 |
| E |
V |
D |
V |
EVDV |
64.64 |
60.42 |
69.98 |
| Q |
S |
W |
V |
QSWV |
65.40 |
70.08 |
20.10 |
| E |
S |
W |
L |
ESWL |
65.65 |
32.39 |
12.96 |
| E |
T |
D |
V |
ETDV |
65.75 |
19.34 |
10.13 |
| R |
T |
W |
V |
RTWV |
65.95 |
63.58 |
34.12 |
| E |
R |
W |
V |
ERWV |
66.25 |
73.54 |
84.36 |
| E |
K |
W |
V |
EKWV |
69.62 |
78.10 |
78.21 |
| E |
T |
M |
V |
ETMV |
70.02 |
42.52 |
11.79 |
| K |
T |
W |
V |
KTWV |
70.41 |
72.01 |
39.02 |
| V |
S |
W |
V |
VSWV |
72.81 |
53.22 |
19.13 |
| H |
S |
W |
V |
HSWV |
73.11 |
73.48 |
21.78 |
| T |
S |
W |
V |
TSWV |
73.42 |
59.63 |
31.54 |
| E |
E |
W |
V |
EEWV |
76.83 |
50.84 |
65.29 |
| E |
N |
W |
V |
ENWV |
77.36 |
73.14 |
77.07 |
| E |
G |
W |
V |
EGWV |
77.80 |
77.50 |
96.96 |
| E |
T |
H |
V |
ETHV |
79.87 |
39.20 |
11.76 |
| E |
T |
R |
V |
ETRV |
80.49 |
34.19 |
7.30 |
| E |
I |
A |
V |
EIAV |
82.18 |
94.10 |
59.51 |
| D |
T |
W |
I |
DTWI |
83.02 |
55.74 |
47.59 |
| F |
S |
W |
V |
FSWV |
83.61 |
69.96 |
29.60 |
| D |
T |
F |
L |
DTFL |
88.62 |
66.62 |
68.98 |
| E |
D |
W |
V |
EDWV |
89.77 |
63.58 |
72.87 |
| I |
S |
W |
V |
ISWV |
91.56 |
62.03 |
32.56 |
| E |
T |
W |
T |
ETWT |
92.32 |
81.00 |
47.53 |
| N |
S |
W |
V |
NSWV |
93.43 |
85.68 |
28.01 |
| S |
T |
D |
V |
STDV |
93.76 |
79.00 |
19.60 |
| E |
T |
P |
V |
ETPV |
96.06 |
36.10 |
16.40 |
| E |
P |
W |
V |
EPWV |
97.08 |
84.84 |
97.77 |
| D |
T |
W |
L |
DTWL |
99.52 |
31.83 |
38.82 |
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Reference:
Urs Wiedemann and Prisca Boisguerin, Rainer Leben, Dietmar Leitner, Gerd Krause, Karin Moelling, Rudolf Volkmer-Engert and Hartmut Oschkinat (2004) submitted.
Last modified: Sun May 02 19:09:10 W. Europe Daylight Time 2004
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